Download Receptor Chemistry Towards the Third Millennium by M. Gianella, G. Marucci, W. Quaglia, U. Gulini PDF

By M. Gianella, G. Marucci, W. Quaglia, U. Gulini

Receptor Chemistry in the direction of the 3rd Millennium is the results of papers offered on the twelfth Camerino-Noordwijkerhout Symposium, held in Camerino, Italy in September 1999. even if a lot is understood in regards to the manner ligands engage with receptors, that have now been remoted, characterised and cloned, many facets nonetheless stay to be explored. specifically, differentiation into special subpopulations and the multiplicity of transduction strategies provide extra particular goals within the look for new drugs.

This e-book may be of curiosity to medicinal chemists, pharmacologists, biochemists and neurologists and also will be a important resource of reference for clinical scholars and postgraduate scholars in similar fields.

Show description

By M. Gianella, G. Marucci, W. Quaglia, U. Gulini

Receptor Chemistry in the direction of the 3rd Millennium is the results of papers offered on the twelfth Camerino-Noordwijkerhout Symposium, held in Camerino, Italy in September 1999. even if a lot is understood in regards to the manner ligands engage with receptors, that have now been remoted, characterised and cloned, many facets nonetheless stay to be explored. specifically, differentiation into special subpopulations and the multiplicity of transduction strategies provide extra particular goals within the look for new drugs.

This e-book may be of curiosity to medicinal chemists, pharmacologists, biochemists and neurologists and also will be a important resource of reference for clinical scholars and postgraduate scholars in similar fields.

Show description

Read or Download Receptor Chemistry Towards the Third Millennium PDF

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Stereochemically-defined lobeline analogues: inhibition of [3H]dopamine uptake and [3H]nicotine binding in rat striatum. Abstracts, College on Problems of Drug Dependence meeting, Acapulco, Mexico, June 12-17, 1999, p. 29. , 1997. Pharmacology of lobeline, a nicotinic receptor ligand. J. Pharmacol. Exp. Ther. 282, 410-419. , 1997. [125I]IPH, an epibatidine analog, binds with high affinity to neuronal nicotinic cholinergic receptors. J. Pharmacol. Exp. Ther. 282, 445-451. , 1995. Characterization of a series of anabaseine-derived compounds reveals that the 3-(4)-dimethylamino-cinnamylidine derivative is a selective agonist at neuronal nicotinic OL7/125I-oLbungarotoxin receptor subtypes.

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